Synthesis and antimicrobial activity of some 1, 2, 4-triazole-3-mercaptoacetic acid derivatives

N Ulusoy, A Gürsoy, G Ötük - Il Farmaco, 2001 - Elsevier
Ethyl 5-(2-furyl)-4-ethyl-1, 2, 4-triazole-3-mercaptoacetate (2), 5-(2-furyl)-4-ethyl-1, 2, 4-
triazole-3-mercaptoacetic acid hydrazide (3) and a series of new N-alkylidene/arylidene-5-(2 …

Design, synthesis, characterization and antimicrobial evaluation of some novel hydrazinecarbothioamide, 4‐thiazolidinone and 1, 2, 4‐triazole‐3‐thione derivatives

ED Dincel, N Ulusoy‐Güzeldemirci… - Journal of …, 2021 - Wiley Online Library
A series of novel hydrazinecarbothioamide (5a, c, f), 4‐thiazolidinone (6a‐e), and 1, 2, 4‐
triazole‐3‐thione (7a‐d) were designed and synthesized. The structural elucidations of the …

[HTML][HTML] Synthesis and antimicrobial activity of new 4-thiazolidinone derivatives containing 2-amino-6-methoxybenzothiazole

NB Patel, FM Shaikh - Saudi Pharmaceutical Journal, 2010 - Elsevier
A novel series of Schiff bases 5a–j and 4-thiazolidinones 6a–j have been prepared from the
building blocks 2-chloro pyridine-3-carboxylic acid [1] and 2-amino-6-methoxy …

[PDF][PDF] Synthesis, characterization and screening of antimicrobial, antituberculosis, antiviral and anticancer activity of novel 1, 3-thiazolidine-4-ones derived from 1-[2 …

E Tatar, İ Küçükgüzel, E De Clercq, F Şahin… - Arkivoc, 2008 - arkat-usa.org
The enhanced prevalence of infectious diseases threatens world population. Although
tuberculosis appeared as a curable disease for years, it is regaining importance due to the …

Synthesis, anticancer activity, and molecular modeling of etodolac‐thioether derivatives as potent methionine aminopeptidase (type II) inhibitors

I Çoruh, Ö Çevik, K Yelekçi, T Djikic… - Archiv der …, 2018 - Wiley Online Library
Abstract A series of (R, S)‐1‐{[5‐(substituted) sulfanyl‐4‐substituted‐4H‐1, 2, 4‐triazole‐3‐
yl] methyl}‐1, 8‐diethyl‐1, 3, 4, 9‐tetrahydropyrano [3, 4‐b] indoles (5a–v) were designed …

Novel 1, 2, 4-triazoles derived from Ibuprofen: synthesis and in vitro evaluation of their mPGES-1 inhibitory and antiproliferative activity

B Bülbül, K Ding, CG Zhan, G Çiftçi, K Yelekçi… - Molecular Diversity, 2023 - Springer
Some novel triazole-bearing ketone and oxime derivatives were synthesized from Ibuprofen.
In vitro cytotoxic activities of all synthesized molecules against five cancer lines (human …

Synthesis, structure, and antifungal evaluation of some novel 1, 2, 4-triazolylmercaptoacetylthiosemicarbazide and 1, 2, 4-triazolylmercaptomethyl-1, 3, 4-thiadiazole …

N Terzioğlu Klip, G Çapan, A Gürsoy… - Journal of Enzyme …, 2010 - Taylor & Francis
Novel 1-[[4-(4-bromophenyl)-5-(2-furyl)-4 H-1, 2, 4-triazole-3-yl] mercaptoacetyl]-4-alkyl/aryl-
3-thiosemicarbazides (5–12) were synthesized by the reaction of 4-(4-bromophenyl)-5-(2 …

Synthesis and antimicrobial evaluation of new 3-alkyl/aryl-2-[((α, α-diphenyl-α-hydroxy) acetyl) hydrazono]-5-methyl-4-thiazolidinones

NU Güzeldemirci, E Ilhan, Ö Küçükbasmaci… - Archives of pharmacal …, 2010 - Springer
New 4-thiazolidinone derivatives of benzilic acid (α, α-diphenyl-α-hydroxyacetic acid) have
been synthesized and evaluated for antibacterial and antifungal activities. The reaction of 1 …

Synthesis, characterization and antimicrobial evaluation of new 2-(2-thienylcarbonyl) hydrazono-3-alkyliaryl-4-thiazolidinone and 2-aryl-3-(2-thienylcarbonyl) amino-4 …

E Dincel, D Satana, S Özbey… - Journal of Research …, 2022 - avesis.hacettepe.edu.tr
A series of novel 2-(2-thienylcarbonyl) hydrazono-3-alkyl/aryl-4-thiazolidinone (2a-f), 2-(2-
thienyl)-5-[(4-bromophenyl) amino]-1, 3, 4-oxadiazole (3), 2-aryl-3-(2-thienylcarbonyparnino …

Synthesis, characterization, and evaluation of antimicrobial activity of Some 1, 2, 4-Triazole derivatives bearing an antipyryl moiety

N Ulusoy, Ö Ateş, Ö Küçükbasmacı, M Kiraz… - Monatshefte für Chemie …, 2003 - Springer
Some novel 4-[[2-[[5-(2-furanyl)-4-alkyl/aryl-4 H-1, 2, 4-triazol-3-yl] thio]-acetyl/propionyl]-
amino]-1, 5-dimethyl-3-oxo-2-phenyl-2, 3-dihydro-1 H-pyrazoles were synthesized and …