1H-Pyrazolo[3,4-b]pyridines: Synthesis and Biomedical Applications

A Donaire-Arias, AM Montagut, R Puig de la Bellacasa… - Molecules, 2022 - mdpi.com
Pyrazolo [3, 4-b] pyridines are a group of heterocyclic compounds presenting two possible
tautomeric forms: the 1 H-and 2 H-isomers. More than 300,000 1 H-pyrazolo [3, 4-b] …

Recent advances in catalytic synthesis of pyridine derivatives

M Torabi, M Yarie, S Baghery, MA Zolfigol - Recent Developments in the …, 2023 - Elsevier
In recent years, the fundamental variety and biological influence of pyridine and its
derivatives make them fascinating aims for preparation. These versatile compounds can be …

Switchable Chemoselectivity in [3 + 3] Annulation of β,γ-Unsaturated α-Ketoesters and 1H-Pyrazol-5-amines by Cooperative Acid Catalysis with NiII and InI

M Tang, M Wang, S Li, C Guo, R Song, D Yang… - Organic …, 2024 - ACS Publications
The exchange of the metal ion from Ni (II) to In (I) leads to a switch in the chemoselectivity of
the [3+ 3] annulation of β, γ-unsaturated α-ketoesters and 1 H-pyrazol-5-amines in the …

Modular and selective synthesis of pyrazolo-azepino-centred polycyclic aromatic and non-aromatic architectures

T Chen, JT Ma, XL Chen, Y Zhou, ZC Yu… - Organic Chemistry …, 2023 - pubs.rsc.org
The pyrazolo-azepino-centred polyheterocyclic fused system is a privileged scaffold, but it
lacks an effective synthetic approach, with modular synthesis being even more scarce …

Heterocyclizations of β-alkoxy, β-diaminoalkyl, and related β-functionalized enones (enals) with NCN-binucleophiles

BV Vashchenko, OO Grygorenko… - Ukrainica Bioorganica …, 2022 - bioorganica.com.ua
This review provides a detailed survey of the present literature data on β-alkoxyvinyl-and β-
enaminocarbonyl compounds as CCC bis-electrophiles in reactions with the common NCN …

Synthesis and reactions of novel imidazo [4, 5-b] pyridine building blocks

TF Dubina, AV Kosarevych, OV Kucher… - Chemistry of …, 2024 - Springer
The synthesis of a novel imidazo [4, 5-b] pyridine and its partially saturated derivative relied
on Michael addition of 1-methyl-1H-imidazol-4-amine to fumaric/maleic or acetylene …

Divergent Synthesis of Isoxazolo[5,4‐b]pyridines

M Li, W Li, M Huang, X Zhang - European Journal of Organic …, 2024 - Wiley Online Library
Isoxazolopyridines are highly significant for the development of pharmaceuticals and new
materials. In continuation of our ongoing research on transformations of 5‐aminoisoxazoles …

Divergent Synthesis of Novel 3 (5)‐Aminoazole–Benzopyrone Hybrids and their Evaluation as α‐Glucosidase Inhibitors

AS Myshko, GP Mrug, SP Bondarenko… - ChemMedChem - Wiley Online Library
An efficient approach has been developed for the trapping in situ generated benzopyrone‐
based ortho‐quinone methide intermediates by 3‐and 5‐amino pyrazoles or isoxazoles. In …

Особливості взаємодії 3-R-ізоксазол-5-амінів з діетил-2-оксосукцинатом. Синтез етил 6-гідрокси-3-R-[1, 2] оксазоло [5, 4-b] піридин-4-карбоксилатів

СВ Толкунов, АС Толкунов, ОВ Смирнова… - Фізико-органічна …, 2021 - er.knutd.edu.ua
Доступність ізоксазоло [5, 4-b] піридинів, які легко одержуються з 5-аміноізоксазолів
реакціями Комба і Дебнера, а також їх різноманітна біоактивність робить цей клас …

[引用][C] СИНТЕЗ ФУНКЦІОНАЛІЗОВАНИХ АНЕЛЬОВАНИХ ПІРИДИНІВ [3+ 3] ГЕТЕРОЦИКЛІЗАЦІЄЮ α-НЕЗАМІЩЕНИХ АМІНОГЕТЕРОЦИКЛІВ ЯК CCN …

АО Толмачов - 2021 - … національний університет імені …