Selective electrophilic di-and monofluorinations for the synthesis of 4-difluoromethyl and 4-fluoromethyl quinazolin (thi) ones by a Selectfluor-triggered multi …
R Zhang, R Ma, Q Fu, R Chen, Z Wang… - Organic Chemistry …, 2022 - pubs.rsc.org
A simple and efficient domino protocol for the selective synthesis of 4-difluoromethyl and 4-
fluoromethyl quinazolin (thi) ones was established from readily available 2 …
fluoromethyl quinazolin (thi) ones was established from readily available 2 …
Synthesis and antimycobacterial activities of some new thiazolylhydrazone derivatives
K Ozadali, OU Tan, P Yogeeswari… - Bioorganic & medicinal …, 2014 - Elsevier
This Letter reports the synthesis and evaluation of some thiazolylhydrazone derivatives for
their in vitro antimycobacterial activities against Mycobacterium tuberculosis H37Rv. The …
their in vitro antimycobacterial activities against Mycobacterium tuberculosis H37Rv. The …
Hydrazone, amide, carbamate, macromolecular and other prodrugs of doxorubicin
S Rollas, G Küçükgüzel - The Open Drug Delivery Journal, 2008 - benthamopen.com
Hydrazone, Amide, Carbamate, Macromolecular and Other Prodrugs of Doxorubicin Page 1
The Open Drug Delivery Journal, 2008, 2, 77-85 77 1874-1266/08 2008 Bentham Open Open …
The Open Drug Delivery Journal, 2008, 2, 77-85 77 1874-1266/08 2008 Bentham Open Open …
[HTML][HTML] Some new hydrazone derivatives bearing the 1, 2, 4-triazole moiety as potential antimycobacterial agents
Objectives: The aim of this study was to synthesize, characterize, and screen some new 1-(4-
((2-(4-substitutedphenyl) hydrazono) methyl) phenyl)-1H-1, 2, 4-triazole derivatives for their …
((2-(4-substitutedphenyl) hydrazono) methyl) phenyl)-1H-1, 2, 4-triazole derivatives for their …
[PDF][PDF] In Vivo Metabolism in Preclinical Drug Development
S Rollas - Preclinical Development Handbook: ADME and …, 2008 - academia.edu
23.2 In Vivo Metabolism of Drug Candidates 23.2. 1 Isolation and Identification of
Metabolites 23.2. 2 Synthesis of Metabolites 23.2. 3 Protein Binding of Metabolites 23.2. 4 …
Metabolites 23.2. 2 Synthesis of Metabolites 23.2. 3 Protein Binding of Metabolites 23.2. 4 …