Structural activity relationship and importance of benzothiazole derivatives in medicinal chemistry: A comprehensive review

M Bhat, SL Belagali - Mini-Reviews in Organic Chemistry, 2020 - ingentaconnect.com
Benzothiazole (1, 3-benzothiazole) is one of the heterocyclic compounds, which is a weak
base having varied biological activities. The unique methine center present in the thiazole …

Recent advances in quantitative structure–activity relationship models of antimalarial drugs

PK Ojha, V Kumar, J Roy, K Roy - Expert Opinion on Drug …, 2021 - Taylor & Francis
Introduction Due to emerging resistance to the first-line artemisinin-based antimalarials and
lack of efficient vaccines and limited chemotherapeutic alternatives, there is an urgent need …

Thiazolidin-4-ones as potential antimicrobial agents: Experimental and in silico evaluation

C Tratrat, A Petrou, A Geronikaki, M Ivanov, M Kostić… - Molecules, 2022 - mdpi.com
Herein, we report computational and experimental evaluations of the antimicrobial activity of
twenty one 2, 3-diaryl-thiazolidin-4-ones. All synthesized compounds exhibited an …

[PDF][PDF] Synthesis and structural profile analysis of the MgO nanoparticles produced through the sol-gel method followed by annealing process

IW Sutapa, AW Wahab, P Taba… - Oriental Journal of …, 2018 - pdfs.semanticscholar.org
MgO nanoparticle was synthesized by sol-gel method from magnesium acetate and oxalic
acid dissolved in methanol followed by annealed process. Characterization of functional …

Dislocation, crystallite size distribution and lattice strain of magnesium oxide nanoparticles

IW Sutapa, A Wahid Wahab, P Taba… - Journal of Physics …, 2018 - iopscience.iop.org
The oxide of magnesium nanoparticles synthesized using sol-gel method and analysis of
the structural properties was conducted. The functional groups of nanoparticles has been …

Pyrazole Schiff base hybrids as anti-malarial agents: synthesis, in vitro screening and computational study

S Aggarwal, D Paliwal, D Kaushik… - … chemistry & high …, 2018 - ingentaconnect.com
Background: Malaria is one of the most vital infectious diseases caused by protozoan
parasites of the Plasmodium genus. As P. falciparum, the cause of most of the severe cases …

[PDF][PDF] Bio-synthesis of gold nanoparticles through bioreduction using the aqueous extract of Muntingia calabura L. leaf

AW Wahab, A Karim, IW Sutapa - Oriental Journal of Chemistry, 2018 - researchgate.net
One of the plants with many functions as tradisional drug is Muntingia calabura L. leaves. It
caused the leaves has high content of tannins, saponins and flavonoids. The presence of …

[PDF][PDF] Aj csian ournalof hemistry aj csian ournalof hemistry

VK SHARMA, A BARDE, S RATTAN - Asian Journal of Chemistry, 2020 - academia.edu
Novel thiazolidine-2, 4-dione (TZD) based pyrimidine derivatives have been synthesized by
Knoevenagel condensation reaction between thiazolidine-2, 4-dione and amino pyrimidinyl …

A quantitative structure-activity relationship approach to determine biotoxicity of amide herbicides for ecotoxicological risk assessment

K Wang, Y Lv, M He, L Tian, F Nie, Z Shao… - Archives of …, 2023 - Springer
Amide herbicides have been widely applied in agriculture and found to be widespread and
affect nontarget organisms in the environment. To better understand the biotoxicity …

Benzothiazole and chromone derivatives as potential ATR kinase inhibitors and anticancer agents

M Frasinyuk, D Chhabria, V Kartsev, H Dilip… - Molecules, 2022 - mdpi.com
Despite extensive studies and the great variety of existing anticancer agents, cancer
treatment remains an aggravating and challenging problem. Therefore, the development of …