The review highlights the hydantoin syntheses presented from the point of view of the
preparation methods. Novel synthetic routes to various hydantoin structures, the advances …

Here, we report a novel “CyClick” strategy for the macrocyclization of peptides that works in
an exclusively intramolecular fashion thereby precluding the formation of dimers and …

A novel base-promoted [3+ 2] cycloaddition reaction of azaoxyallyl cations with hexahydro-
1, 3, 5-triazines has been developed, affording 4-imidazolidinones in moderate to good …

An Et3N-catalyzed cascade [3+ 2]-annulation of β-oxo-acrylamides with cyclic N-sulfonyl
ketimines or sulfamate-derived imines is developed under mild reaction conditions, which …

Despite the importance of the 4-imidazolidinone scaffold in bioactive compounds or
organocatalysts, methodologies to access these nitrogenated heterocycles remain scarce …

An efficient regio-and diastereoselective cyclization of sulfamate-derived cyclic imines with
unsubstituted or monosubstituted α-halo hydroxamates is developed under mild conditions …

The moiety of 4-imidazolidinone is an important structural motif in organic synthesis and
medicinal chemistry. We present the synthesis of 4-imidazolidinones from various diamides …

Aiming to develop novel anticonvulsant agents a new series of novel
cycloalkanecarboxamide parabanic acid hybrids series 8, 9 and 10 possessing the essential …

Abstract A new set of 1, 3-benzodioxoles and 1, 4-benzodioxines was designed and
synthesized starting from gallic acid as anticancer agents. The antiproliferative effect of the …

Herein a novel and robust methodology to spiroimidazolidinones has been developed
under a mild reaction. The reaction of (Z)-2-azido-3-phenylacrylic acids 1, aldehydes 2 …