Piperidines are among the most important synthetic fragments for designing drugs and play
a significant role in the pharmaceutical industry. Their derivatives are present in more than …

Nitrogen-containing heterocycles are among the most significant as they are found in a wide
range of pharmacologically active molecules. Lewis acids are regarded as crucial activation …

Gold-catalyzed 5-exo-dig hydroamination on O-homopropargylic hydroxylamine gave
expeditious access to methylene isoxazolidine. Excess catalyst loading led to facile 1, 3 …

Lewis-acid-catalyzed 5-endo-dig reductive hydroalkoxylation cascade on propargylic N-
hydroxylamine gave expedient, stereoselective access to isoxazolidine derivatives. The …

TMSOTf‐mediated 5‐endo‐dig aminocyclization followed by N‐to C‐[1, 3]‐sulfonyl
migration on N¬‐homopropargyl hydroxylamines gave diastereoselective access to …

Stereoselective syntheses of pyrrolidines and piperidines bearing hydrophobic chains have
been achieved through a metal free, Lewis acid-mediated 5/6-endo-dig reductive …

A copper-catalyzed cascade reaction of diazo compounds with 1, n-allenynes (n= 6, 7) was
reported, which provides efficient access to various functionalized 3-azabicyclo [m. 2.0] …

Fused indolizidines and quinolizidines are important skeletons in a variety of natural
products and pharmacologically important compounds. A one-pot tandem route from amide …

A Lewis acid-mediated, 5/6/7/8-endo-dig reductive hydroalkoxylation cascade on enynols
gives expeditious, diastereoselective access to small and medium ring cyclic ethers with a …

A protocol involving intramolecular formal [4+ 2]‐cycloaddition of in situ generated o‐aza‐
quinone methide for the facile synthesis of 1, 4‐heterocycle‐fused quinoline motifs is …